SCHEMBL25425980

SCHEMBL25425980

COc1cccc(CNCc2ccc(-n3ccnc3)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.53
CYP11B2 P19099 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.51
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
HTT P42858 1/20 0.51
HDAC1 Q13547 2/20 0.50
PDE5A O76074 2/20 0.49
TBXAS1 P24557 2/20 0.49
PDE3B Q13370 2/20 0.49
PDE3A Q14432 2/20 0.49
HDAC3 O15379 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
CHRM2 P08172 1/20 0.48
ADRB1 P08588 2/20 0.47
ADRB2 P07550 1/20 0.47
ADRB3 P13945 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25255599 0.91 CYP11B1 (0.54) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1
SCHEMBL30245596 0.91 CYP11B1 (0.54) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1
SCHEMBL5046565 0.79 MAPT (0.46) SMN1; SMN2KDM4EALDH1A1HTTMEN1
SCHEMBL25426943 0.79 DGAT2 (0.63) SMN1; SMN2KDM4EALDH1A1HTTHDAC1
SCHEMBL6389607 0.78 CYP11B1 (0.71) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1
SCHEMBL30245843 0.78 PDE5A (0.44) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1
SCHEMBL29194699 0.77 CYP11B1 (0.52) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1
SCHEMBL9416628 0.77 KDM4E (0.79) SMN1; SMN2KDM4EALDH1A1HTTHDAC1
SCHEMBL25427024 0.77 CYP11B1 (0.46) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1
SCHEMBL25427086 0.77 CYP11B1 (0.46) CYP11B1CYP11B2SMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4384516-A1 AMINOARYL-INTEGRIN AGONISTS COMPOUNDS Texas Heart Institute (US) 2024-06-19 EP disclosed
CN-117916237-A Amino aryl integrin agonist compounds 德克萨斯心脏研究所 2024-04-19 CN disclosed
WO-2023018472-A9 AMINOARYL-INTEGRIN AGONISTS COMPOUNDS TEXAS HEART INSTITUTE (US) 2023-07-13 WO disclosed
WO-2023018472-A1 AMINOARYL-INTEGRIN AGONISTS COMPOUNDS TEXAS HEART INSTITUTE (US) 2023-02-16 WO disclosed