SCHEMBL25257982

SCHEMBL25257982

Cc1ccccc1S(=O)(=O)n1cc(I)c2cc(Cl)cnc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.47
RAPGEF4 Q8WZA2 1/20 0.40
DRD2 P14416 2/20 0.38
CYP3A4 P08684 1/20 0.38
SLC6A2 P23975 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR7 P34969 1/20 0.38
HRH1 P35367 1/20 0.38
ADRA1B P35368 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KMT2A Q03164 2/20 0.38
HTT P42858 3/20 0.37
TSHR P16473 2/20 0.37
KLK7 P49862 1/20 0.36
POLB P06746 3/20 0.35
DRD1 P21728 1/20 0.35
PIK3C3 Q8NEB9 1/20 0.35
LMNA P02545 1/20 0.34
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25297234 0.86 BRD4 (0.47) BRD4RAPGEF4KMT2AHTTTSHR
SCHEMBL29200258 0.83 DRD2 (0.37) BRD4RAPGEF4DRD2CYP3A4SLC6A2
SCHEMBL1266871 0.83 BRD4 (0.58) BRD4DRD2CYP3A4SLC6A2HTR2A
SCHEMBL25299441 0.81 DRD2 (0.36) BRD4RAPGEF4DRD2CYP3A4SLC6A2
SCHEMBL31150811 0.81 BRD4 (0.51) BRD4RAPGEF4DRD2CYP3A4SLC6A2
SCHEMBL18995268 0.81 BRD4 (0.51) BRD4RAPGEF4DRD2CYP3A4SLC6A2
SCHEMBL25300843 0.79 PIK3C3 (0.36) BRD4RAPGEF4DRD2CYP3A4SLC6A2
SCHEMBL14678605 0.79 CYP3A4 (0.35) BRD4RAPGEF4DRD2CYP3A4SLC6A2
SCHEMBL25302927 0.75 HPGD (0.41) BRD4KMT2AHTTTSHRLMNA
SCHEMBL28769144 0.74 BRD4 (0.44) BRD4RAPGEF4HTTTSHRPIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed