SCHEMBL25258958

SCHEMBL25258958

CCOC(=O)c1cc(OC)c2c(c1)nc(N)n2Cc1ccc(Br)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
CASP1 P29466 2/20 0.44
CASP7 P55210 2/20 0.44
HSD17B10 Q99714 2/20 0.44
USP2 O75604 1/20 0.44
GLA P06280 1/20 0.44
MAPK1 P28482 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
STING1 Q86WV6 1/20 0.42
TYMS P04818 1/20 0.42
ENPP1 P22413 2/20 0.42
TSHR P16473 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HSD17B2 P37059 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30586455 1.00 GAA (0.44) GAAKDM4EALDH1A1HPGDCASP1
SCHEMBL25262670 0.90 SMN1; SMN2 (0.44) GAAKDM4EALDH1A1HPGDCASP1
SCHEMBL30586457 0.90 SMN1; SMN2 (0.44) GAAKDM4EALDH1A1HPGDCASP1
SCHEMBL30586478 0.87 CA2 (0.44) GAAKDM4EALDH1A1HPGDCASP1
SCHEMBL25257071 0.87 CA2 (0.44) GAAKDM4EALDH1A1HPGDCASP1
SCHEMBL29036924 0.80 HSD17B2 (0.39) KDM4EALDH1A1HPGDMAPK1STING1
SCHEMBL25253344 0.78 CA2 (0.43) ALDH1A1USP2NPSR1TSHRLMNA
SCHEMBL30586476 0.78 CA2 (0.43) ALDH1A1USP2NPSR1TSHRLMNA
SCHEMBL25826736 0.78 ENPP1 (0.70) STING1ENPP1
SCHEMBL25259879 0.78 STING1 (0.47) STING1ENPP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116444544-A Benzimidazole compound and medical application thereof 中国科学院上海药物研究所 2023-07-18 CN disclosed
WO-2023131333-A1 BENZIMIDAZOLE COMPOUND AND MEDICAL USE THEREOF 中国科学院上海药物研究所 2023-07-13 WO disclosed
WO-2023131333-A1 BENZIMIDAZOLE COMPOUND AND MEDICAL USE THEREOF 中国科学院上海药物研究所 2023-07-13 WO disclosed