SCHEMBL25284302

SCHEMBL25284302

CCOC(=O)c1cnc(N(C)CCN(C)C)nc1C#C[Si](C(C)C)(C(C)C)C(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
HSD17B10 Q99714 1/20 0.39
POLB P06746 2/20 0.39
RAD52 P43351 2/20 0.39
KMT2A Q03164 2/20 0.38
UHRF1 Q96T88 1/20 0.38
HSP90AA1 P07900 1/20 0.37
JUN P05412 2/20 0.36
NFKB1 P19838 2/20 0.36
NFKB2 Q00653 2/20 0.36
RELA Q04206 2/20 0.36
KDM4E B2RXH2 2/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TP53 P04637 1/20 0.36
ALOX15 P16050 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HCRTR1 O43613 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25241696 0.86 SYK (0.38) ALDH1A1HSD17B10KDM4EALOX15HCRTR1
SCHEMBL31140700 0.86 SYK (0.38) ALDH1A1HSD17B10KDM4EALOX15HCRTR1
SCHEMBL25288509 0.85 SYK (0.46) HCRTR1HCRTR2SYK
SCHEMBL31140646 0.85 SYK (0.46) HCRTR1HCRTR2SYK
SCHEMBL25239216 0.77 ALDH1A1 (0.46) ALDH1A1HSD17B10POLBRAD52KMT2A
SCHEMBL31140705 0.77 ALDH1A1 (0.46) ALDH1A1HSD17B10POLBRAD52KMT2A
SCHEMBL25284311 0.76 KDM4E (0.49) ALDH1A1HSD17B10POLBRAD52KMT2A
SCHEMBL5071189 0.73 KDM4E (0.64) ALDH1A1HSD17B10POLBRAD52HSP90AA1
SCHEMBL6984025 0.70 KDM5B (0.44) ALDH1A1HSD17B10POLBJUNNFKB1
SCHEMBL6982223 0.67 CYP1A2 (0.50) ALDH1A1POLBKMT2AKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118525018-A Bialkyne compound and application thereof 上海艾力斯医药科技股份有限公司 2024-08-20 CN disclosed
WO-2023116779-A1 DIALKYNE COMPOUND AND USE THEREOF 上海艾力斯医药科技股份有限公司 2023-06-29 WO disclosed