SCHEMBL6984025

SCHEMBL6984025

CCOC(=O)c1cnc(N(C)CCN(C)C)nc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 2/20 0.44
KDM5A P29375 1/20 0.44
KDM5C P41229 1/20 0.44
KDM4C Q9H3R0 1/20 0.44
ALDH1A1 P00352 6/20 0.43
MAPT P10636 2/20 0.43
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA7 P43166 2/20 0.40
CA9 Q16790 2/20 0.40
CA14 Q9ULX7 2/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
HSD17B10 Q99714 2/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24925656 0.87 ALDH1A1 (0.41) ALDH1A1MAPTCYP2C9CYP2C19CA12
SCHEMBL11530672 0.82 ALDH1A1 (0.56) ALDH1A1MAPTCYP2C9CYP2C19CA12
SCHEMBL31140705 0.79 ALDH1A1 (0.46) ALDH1A1MAPTHSD17B10NPC1RAB9A
SCHEMBL25239216 0.79 ALDH1A1 (0.46) ALDH1A1MAPTHSD17B10NPC1RAB9A
SCHEMBL6982188 0.79 ALDH1A1 (0.61) KDM5BKDM5AKDM5CALDH1A1MAPT
SCHEMBL31141612 0.79 RAB9A (0.42) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL25284311 0.78 KDM4E (0.49) ALDH1A1HSD17B10NPC1RAB9ACYP1A2
SCHEMBL24218501 0.77 LMNA (0.42) ALDH1A1MAPTHSD17B10NPC1RAB9A
SCHEMBL24925660 0.77 CKS1B (0.48) ALDH1A1MAPTCA12CA1CA2
SCHEMBL6982223 0.75 CYP1A2 (0.50) KDM5BKDM5AKDM5CKDM4CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1093367-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-03-05 EP claimed
EP-1093367-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-25 EP claimed
WO-1999066925-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-29 WO claimed
EP-1093367-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-03-05 EP disclosed
EP-1093367-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-25 EP disclosed
WO-1999066925-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1999-12-29 WO disclosed