SCHEMBL25303151

SCHEMBL25303151

CC(C)(O)C(=O)N1CCc2cc(Cl)cc(C3COCCN3)c2C1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.35
ESR1 P03372 2/20 0.34
ESR2 Q92731 2/20 0.34
PIK3R1 P27986 4/20 0.32
PIK3CA P42336 4/20 0.32
SLC18A2 Q05940 2/20 0.31
PDK2 Q15119 1/20 0.31
BAZ2B Q9UIF8 1/20 0.31
NAMPT P43490 2/20 0.30
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25302877 1.00 RIPK1 (0.35) RIPK1ESR1ESR2PIK3R1PIK3CA
SCHEMBL25838463 0.89 RIPK1 (0.34) RIPK1ESR1ESR2PIK3R1PIK3CA
SCHEMBL30491452 0.89 BAZ2B (0.39) BAZ2B
SCHEMBL30491431 0.85 AKR1C3 (0.33) BAZ2B
SCHEMBL25305291 0.85 AKR1C3 (0.36) DRD2DRD3
SCHEMBL25305296 0.85 AKR1C3 (0.36) DRD2DRD3
SCHEMBL25303656 0.83 CGAS (0.46) SLC18A2NAMPT
SCHEMBL30491427 0.83 PRMT5 (0.33) PIK3CADRD2DRD3
SCHEMBL25299917 0.83
SCHEMBL25303659 0.83 CGAS (0.46) SLC18A2NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed
WO-2022184152-A1 FUSED RING SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2022-09-09 WO disclosed