SCHEMBL25307184

SCHEMBL25307184

COC1CO[C@H](COCc2ccccc2)C1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
TAAR1 Q96RJ0 1/20 0.43
TSHR P16473 2/20 0.40
BACE1 P56817 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
HRH4 Q9H3N8 4/20 0.39
HRH3 Q9Y5N1 4/20 0.39
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSK P43235 1/20 0.38
PTPN1 P18031 1/20 0.38
CDC25B P30305 1/20 0.38
DRD1 P21728 1/20 0.38
CYP3A4 P08684 3/20 0.36
MAPT P10636 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25306201 0.87 LMNA (0.45) LMNATAAR1TSHRL3MBTL1HRH4
SCHEMBL25307033 0.87 LMNA (0.45) LMNATAAR1TSHRL3MBTL1HRH4
SCHEMBL23278064 0.87 LMNA (0.47) LMNATAAR1TSHRBACE1HRH4
SCHEMBL1564320 0.86 LMNA (0.44) LMNATAAR1TSHRBACE1L3MBTL1
SCHEMBL1565954 0.86 LMNA (0.44) LMNATAAR1TSHRBACE1L3MBTL1
SCHEMBL24982368 0.83 LMNA (0.48) LMNATAAR1TSHRL3MBTL1HRH4
SCHEMBL29295670 0.80 LMNA (0.45) LMNATAAR1HRH4HRH3BCHE
SCHEMBL11556022 0.79 CTSL (0.43) HRH3CTSLCTSBCTSKMAPT
SCHEMBL715660 0.79 LMNA (0.57) LMNATAAR1TSHRHRH4HRH3
SCHEMBL306297 0.79 LMNA (0.57) LMNATAAR1TSHRHRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260028356-A1 1,3,4,7-TETRAHYDRO-2H-PYRROLO[3',2':5,6]PYRIDO[2,3-B][1,4]OXAZEPINE BCL-2 INHIBITORS ABBVIE INC (US) 2026-01-29 US disclosed
US-20250066388-A1 1,3,4,7-TETRAHYDRO-2H-PYRROLO[3',2':5,6]PYRIDO[2,3-B][1,4]OXAZEPINE BCL-2 INHIBITORS ABBVIE INC (US) 2025-02-27 US disclosed
CN-119053610-A 1,3,4, 7-Tetrahydro-2H-pyrrolo [3',2':5,6] pyrido [2,3-b ] [1,4] oxazepine Bcl-2 inhibitors 艾伯维公司 2024-11-29 CN disclosed
US-11964990-B2 1,3,4,7-tetrahydro-2H-pyrrolo[3′,2′:5,6]pyrido[2,3-b][1,4]oxazepine bcl-2 inhibitors ABBVIE INC. (US) 2024-04-23 US disclosed
US-20230234971-A1 1,3,4,7-Tetrahydro-2H-pyrrolo[3',2':5,6]pyrido[2,3-b][1,4]oxazepine Bcl-2 Inhibitors ABBVIE INC. (US) 2023-07-27 US disclosed
WO-2023141536-A1 1,3,4,7-TETRAHYDRO-2H-PYRROLO [3',2':5,6] PYRIDO[2,3-B] [1,4] OXAZEPINE BC1-2 INHIBITORS ABBVIE INC. (US) 2023-07-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260028356-A1 1,3,4,7-TETRAHYDRO-2H-PYRROLO[3',2':5,6]PYRIDO[2,3-B][1,4]OXAZEPINE BCL-2 INHIBITORS BCL9L, BCL2L2, BCL2L1 LMNA 1548/4885TAAR1 2001/4885TSHR 2171/4885
US-20250066388-A1 1,3,4,7-TETRAHYDRO-2H-PYRROLO[3',2':5,6]PYRIDO[2,3-B][1,4]OXAZEPINE BCL-2 INHIBITORS BCL9L, BCL2L1, BCL2L2 LMNA 975/4885TAAR1 2721/4885TSHR 2736/4885
US-20230234971-A1 1,3,4,7-Tetrahydro-2H-pyrrolo[3',2':5,6]pyrido[2,3-b][1,4]oxazepine Bcl-2 Inhibitors BCL9L, BCL2L1, BCL2L2 LMNA 975/4885TAAR1 2721/4885TSHR 2736/4885
US-11964990-B2 1,3,4,7-tetrahydro-2H-pyrrolo[3′,2′:5,6]pyrido[2,3-b][1,4]oxazepine bcl-2 inhibitors BCL9L, BCL2L1, BCL9 LMNA 964/4885TAAR1 2736/4885TSHR 2721/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.