SCHEMBL25307190

SCHEMBL25307190

CCOC(=O)c1nn(Cc2ccc(OC)cc2)c(=O)c2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
PKM P14618 2/20 0.58
GAA P10253 1/20 0.58
MAPT P10636 2/20 0.53
LMNA P02545 3/20 0.52
HTT P42858 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
AURKA O14965 1/20 0.52
AURKB Q96GD4 1/20 0.52
POLB P06746 1/20 0.52
KMT2A Q03164 4/20 0.51
MEN1 O00255 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
ELANE P08246 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16377892 0.84 PTGER4 (0.56) ALDH1A1MAPTPOLBKMT2AMEN1
SCHEMBL9925003 0.82 PTGDR2 (0.54) ALDH1A1GAAMAPTLMNAL3MBTL1
SCHEMBL22609303 0.80 PDE4D (0.53) ALDH1A1GAAMAPTLMNAL3MBTL1
SCHEMBL25309590 0.80 ALDH1A1 (0.64) ALDH1A1PKMGAAMAPTLMNA
SCHEMBL12933531 0.79 ALDH1A1 (0.56) ALDH1A1PKMGAALMNAPOLB
SCHEMBL25313395 0.78 ALDH1A1 (0.55) ALDH1A1PKMGAAHTTAURKA
SCHEMBL19402534 0.78 ELANE (0.56) ELANE
SCHEMBL3793270 0.78 MAPT (0.51) ALDH1A1GAAMAPTHTTL3MBTL1
SCHEMBL16244384 0.78 MAPT (0.51) ALDH1A1PKMGAAMAPTKMT2A
SCHEMBL31409773 0.77 AURKA (0.55) ALDH1A1PKMGAAMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023139536-A1 (4-PIPERAZIN-1YL)-4-ALKYL-PHTHALAZIN-1(2H)-ONE COMPOUNDS AS PARP7 INHIBITORS RHIZEN PHARMACEUTICALS AG (CH) 2023-07-27 WO disclosed