SCHEMBL25308804

SCHEMBL25308804

NC(=O)c1cccnc1N1CCNC(=O)C1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.46
KMT2A Q03164 2/20 0.42
PIK3CA P42336 1/20 0.40
MTOR P42345 1/20 0.40
TRPV1 Q8NER1 1/20 0.39
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
GRIA1 P42261 1/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CHIA Q9BZP6 1/20 0.39
RPS6KB1 P23443 1/20 0.39
PRKCA P17252 1/20 0.39
PRKCQ Q04759 1/20 0.39
PRKCD Q05655 1/20 0.39
PRKCH P24723 1/20 0.39
PRKCE Q02156 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4538970 0.83 EPHX2 (0.52) KMT2ATRPV1MEN1CYP1A2CYP3A4
SCHEMBL30945091 0.83 EPHX2 (0.52) KMT2ATRPV1MEN1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL5901187 0.82 EPHX2 (0.51) KMT2ATRPV1MEN1CYP1A2CYP3A4
SCHEMBL14377416 0.80 GRIN2D (0.55) KMT2APIK3CAMTORGRIA1MEN1
SCHEMBL883905 0.78 KMT2A (0.58) PARP1KMT2ATRPV1MEN1CYP1A2
SCHEMBL10094631 0.77 HSD11B1 (0.46) KMT2APIK3CAMTORTRPV1GRIA1
SCHEMBL29574686 0.77 KMT2A (0.44) PARP1KMT2ATRPV1DDB1CRBN
SCHEMBL28189129 0.77 KMT2A (0.60) PARP1KMT2ATRPV1MEN1CYP1A2
SCHEMBL353774 0.74 AURKA (0.60) PARP1KMT2ATRPV1MEN1CYP1A2
SCHEMBL28275410 0.74 CHIA (0.65) PARP1KMT2AMEN1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134708-A1 THIAZOLOPYRIDYL AMIDE DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS BEIGENE , LTD. (KY) 2023-07-20 WO disclosed