SCHEMBL25317776

SCHEMBL25317776

COc1cc(C(F)F)nn1-c1[c]ccc(Cl)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 5/20 0.34
PTGS1 P23219 4/20 0.34
PTGS2 P35354 4/20 0.34
PDE4B Q07343 2/20 0.34
POLB P06746 1/20 0.33
PDE3A Q14432 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25318332 0.83 USP1 (0.32) PTGS1PTGS2KDM4EMEN1ALDH1A1
SCHEMBL25317152 0.80 PTGS1 (0.30) PTGS1PTGS2
SCHEMBL25319788 0.72 SLC34A1 (0.37) MEN1CYP2C9CYP2C19HTTKMT2A
SCHEMBL25949125 0.71 PDE4B (0.42) CASRPTGS1PTGS2PDE4BPOLB
SCHEMBL25319131 0.69
SCHEMBL25320781 0.69
SCHEMBL25320904 0.69 F2RL3 (0.32)
SCHEMBL25320409 0.69 CASR (0.35) CASRPTGS1PTGS2PDE4BPDE3A
SCHEMBL25427261 0.68 PDE4B (0.31) CASRPTGS1PTGS2PDE4BPDE3A
SCHEMBL25318310 0.64 HTT (0.33) MEN1CYP2C9CYP2C19HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023139085-A1 NEW BENZIMIDAZOLE PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2023-07-27 WO disclosed