SCHEMBL25320409

SCHEMBL25320409

COc1cc(C(F)F)nn1-c1nc(Cl)ccc1CC=O

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASR P41180 5/20 0.35
PTGS1 P23219 4/20 0.33
PTGS2 P35354 4/20 0.33
PDE4B Q07343 2/20 0.33
PDE3A Q14432 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25321980 0.86 KDM4E (0.33) PTGS1PTGS2
SCHEMBL25317896 0.84 ALDH1A1 (0.32) PTGS1PTGS2
SCHEMBL25318523 0.83
SCHEMBL25949125 0.77 PDE4B (0.42) CASRPTGS1PTGS2PDE4BPDE3A
SCHEMBL25319677 0.74 HTT (0.34)
SCHEMBL25318412 0.73 HTT (0.46) PTGS2
SCHEMBL25317388 0.73
SCHEMBL25427261 0.72 PDE4B (0.31) CASRPTGS1PTGS2PDE4BPDE3A
SCHEMBL25317254 0.72 MEN1 (0.32)
SCHEMBL25317776 0.69 CASR (0.34) CASRPTGS1PTGS2PDE4BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023139085-A1 NEW BENZIMIDAZOLE PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2023-07-27 WO disclosed