SCHEMBL2531824

SCHEMBL2531824

COc1cc(-c2ccc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)ccc1OCCN1CCNCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 9/20 0.56
KIT P10721 1/20 0.49
LRRK2 Q5S007 2/20 0.47
MAP4K1 Q92918 5/20 0.44
IL2 P60568 2/20 0.44
SGK1 O00141 1/20 0.43
IKBKB O14920 1/20 0.43
AURKA O14965 1/20 0.43
CHUK O15111 1/20 0.43
PRKAB2 O43741 1/20 0.43
ROCK2 O75116 1/20 0.43
ABL1 P00519 1/20 0.43
NTRK1 P04629 1/20 0.43
INSR P06213 1/20 0.43
LCK P06239 1/20 0.43
CDK1 P06493 1/20 0.43
IGF1R P08069 1/20 0.43
MET P08581 1/20 0.43
CYP3A4 P08684 1/20 0.43
SRC P12931 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL721560 0.90 MAP3K11 (0.71) MAP3K11KITLRRK2MAP4K1IL2
SCHEMBL2527600 0.81 MAP3K11 (0.73) MAP3K11KITLRRK2
SCHEMBL7172012 0.78 MAP3K11 (0.53) MAP3K11KITMAPK14LTA4HTLR7
SCHEMBL10164830 0.77 MAP3K11 (0.51) MAP3K11KITLRRK2MAP4K1IL2
SCHEMBL2526092 0.76 MAP3K11 (0.60) MAP3K11KITLRRK2IGF1RCYP3A4
SCHEMBL722011 0.74 KIT (0.56) MAP3K11KITLRRK2MAP4K1IL2
SCHEMBL12763551 0.73 KIT (0.61) KITMAP4K1IL2
SCHEMBL7905848 0.72 KIT (0.60) KITMAP4K1IL2
SCHEMBL2981587 0.72 PRKCQ (0.78)
SCHEMBL721043 0.72 MAP3K11 (1.00) MAP3K11LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379561-A2 MLK INHIBITORS AND METHODS OF USE University Of Rochester (US) 2011-10-26 EP disclosed
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed