SCHEMBL2526092

SCHEMBL2526092

COc1cc(-c2ccc3[nH]cc(-c4ccc5[nH]ccc5c4)c3c2)ccc1N

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 9/20 0.60
LRRK2 Q5S007 2/20 0.56
CYP3A4 P08684 3/20 0.48
CYP2D6 P10635 2/20 0.48
ALDH1A1 P00352 1/20 0.48
TSHR P16473 1/20 0.48
HSD17B10 Q99714 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
CYP2C9 P11712 1/20 0.47
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
HCRTR1 O43613 1/20 0.45
CASP3 P42574 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
KIT P10721 4/20 0.45
PRKCQ Q04759 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2527600 0.89 MAP3K11 (0.73) MAP3K11LRRK2MEN1NPC1HCRTR1
SCHEMBL724259 0.86 MAP3K11 (0.83) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9
SCHEMBL2522333 0.78 MAP3K11 (0.80) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9
SCHEMBL2523833 0.78 MAP3K11 (0.72) MAP3K11CYP3A4CYP2D6ALDH1A1TSHR
SCHEMBL27841169 0.77 MAP3K11 (0.83) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9
SCHEMBL722601 0.77 MAP3K11 (0.58) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9
SCHEMBL2526465 0.77 NPC1 (0.71) MAP3K11LRRK2CYP3A4CYP2D6CYP2C9
SCHEMBL2531824 0.76 MAP3K11 (0.56) MAP3K11LRRK2CYP3A4KITIGF1R
SCHEMBL720862 0.75 MAP3K11 (1.00) MAP3K11LRRK2CYP3A4CYP2D6KIT
SCHEMBL4339872 0.74 MAP3K11 (0.63) MAP3K11LRRK2MEN1NPC1HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379561-A2 MLK INHIBITORS AND METHODS OF USE University Of Rochester (US) 2011-10-26 EP disclosed
WO-2010068483-A2 MLK INHIBITORS AND METHODS OF USE UNIVERSITY OF ROCHESTER (US) 2010-06-17 WO disclosed