SCHEMBL25323326

SCHEMBL25323326

Cc1cc(Br)c2cnn(COCC[Si](C)(C)C)c2n1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.36
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
RECQL P46063 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PNP P00491 2/20 0.32
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30509530 1.00 DGAT1 (0.36) DGAT1MAPTTSHRRECQLNPSR1
SCHEMBL29514198 0.83 DGAT1 (0.36) DGAT1PNP
SCHEMBL30413120 0.78 DGAT1 (0.37) DGAT1MAPTNPC1
SCHEMBL25324687 0.78 DGAT1 (0.37) DGAT1MAPTNPC1
SCHEMBL29514132 0.78 UCHL1 (0.33) MAPTTSHRRECQLNPSR1
SCHEMBL26661569 0.78 UCHL1 (0.33) MAPTTSHRRECQLNPSR1
SCHEMBL26720557 0.78 DGAT1 (0.37) DGAT1PNP
SCHEMBL26720567 0.75 HSP90AA1 (0.36) DGAT1MAPTPNPNPC1
SCHEMBL25875898 0.75 MAPT (0.33) DGAT1MAPTPNP
SCHEMBL24328469 0.75 HSP90AA1 (0.35) DGAT1MAPTPNPNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230339900-A1 CASEIN KINASE 1 DELTA MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2023-10-26 US disclosed
US-20230339900-A1 CASEIN KINASE 1 DELTA MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2023-10-26 US disclosed
US-20230339900-A1 CASEIN KINASE 1 DELTA MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2023-10-26 US disclosed
EP-4214199-A1 CASEIN KINASE 1 DELTA MODULATORS JANSSEN Pharmaceutica NV (BE) 2023-07-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230339900-A1 CASEIN KINASE 1 DELTA MODULATORS CSNK1D, CSNK1A1, CSNK2A1 DGAT1 3673/4885MAPT 364/4885TSHR 2841/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.