SCHEMBL2532974

SCHEMBL2532974

NC(=O)N(c1ccccc1)c1nc(C2CCOCC2)nc(N2CCOCC2)n1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.47
PIK3CA P42336 7/20 0.47
MTOR P42345 7/20 0.47
LMNA P02545 3/20 0.46
TSHR P16473 2/20 0.46
HTT P42858 2/20 0.44
POLB P06746 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GPR55 Q9Y2T6 1/20 0.44
PIK3CD O00329 3/20 0.42
PIK3CB P42338 3/20 0.42
ALDH1A1 P00352 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PIK3CG P48736 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2534195 0.87 PKM (0.56) PKMPIK3CAMTORLMNATSHR
SCHEMBL2532976 0.81 PIK3CA (0.61) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL4455473 0.80 PIK3CA (0.49) PKMPIK3CAMTORLMNATSHR
SCHEMBL2535375 0.79 PIK3CA (0.56) PIK3CAMTORPIK3CDPIK3CBPIK3CG
SCHEMBL2534318 0.77 MTOR (0.43) PKMPIK3CAMTORLMNATSHR
SCHEMBL17773015 0.71 LMNA (0.44) PKMPIK3CAMTORLMNATSHR
SCHEMBL29000061 0.70 PIK3CA (0.64) PIK3CAMTORALDH1A1NPSR1PIK3CG
SCHEMBL9619266 0.70 LMNA (0.52) PKMPIK3CAMTORLMNATSHR
SCHEMBL19665253 0.69 LMNA (0.86) PKMPIK3CAMTORLMNATSHR
SCHEMBL3797375 0.68 PDE4A (0.42) PIK3CAMTORLMNAHTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8039469-B2 Triazine compounds as PI3 kinase and mTOR inhibitors WYETH LLC (US) 2011-10-18 US disclosed