SCHEMBL25335656

SCHEMBL25335656

Fc1cc(Br)cc2[nH]nc(I)c12

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 2/20 0.34
JAK2 O60674 2/20 0.34
GPR17 Q13304 1/20 0.33
DYRK1A Q13627 1/20 0.33
IDO1 P14902 1/20 0.30
TDO2 P48775 1/20 0.30
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29490990 1.00 PDPK1 (0.34) PDPK1JAK2GPR17DYRK1AIDO1
SCHEMBL14738326 0.81 MAP2K4 (0.33) GPR17
SCHEMBL14737657 0.78 TRPA1 (0.35)
SCHEMBL30467571 0.78 PDPK1 (0.34) PDPK1JAK2DYRK1AIDO1TDO2
SCHEMBL31162464 0.78 PDPK1 (0.34) PDPK1JAK2GPR17DYRK1AIDO1
SCHEMBL24252918 0.78 PDPK1 (0.34) PDPK1JAK2DYRK1AIDO1TDO2
SCHEMBL2144129 0.78 PDPK1 (0.34) PDPK1JAK2GPR17DYRK1AIDO1
SCHEMBL1317469 0.78 PDPK1 (0.50) PDPK1JAK2GPR17DYRK1AIDO1
SCHEMBL31393082 0.77 DYRK1A (0.32) PDPK1JAK2DYRK1A
SCHEMBL31313054 0.77 JAK1 (0.33) PDPK1JAK2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122055363-A Compounds and methods for modulating splicing 雷密克斯医疗公司 2026-05-15 CN disclosed
EP-4724438-A1 COMPOUNDS AND METHODS FOR MODULATING SPLICING Remix Therapeutics Inc. (US) 2026-04-15 EP disclosed
WO-2024259015-A1 COMPOUNDS AND METHODS FOR MODULATING SPLICING REMIX THERAPEUTICS INC. (US) 2024-12-19 WO disclosed
US-20240083861-A1 HSD17B13 INHIBITORS AND USES THEREOF FL2022-001, INC. 2024-03-14 US disclosed
EP-4221703-A1 HSD17B13 INHIBITORS AND USES THEREOF FL2022-001, Inc. (US) 2023-08-09 EP disclosed
WO-2022072517-A1 HSD17B13 INHIBITORS AND USES THEREOF METACRINE, INC. (US) 2022-04-07 WO disclosed
CN-113831326-A Condensed heterocyclic derivative and application thereof in medicine 四川海思科制药有限公司 2021-12-24 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240083861-A1 HSD17B13 INHIBITORS AND USES THEREOF HSD17B3, HSD17B11, HSD17B1 PDPK1 1978/4885JAK2 3555/4885GPR17 968/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.