SCHEMBL25339683

SCHEMBL25339683

CC1=C[C@@H](NC(=O)OC(C)(C)C)Cc2c1cc(OCc1ccccc1)c(N(CC(=O)O)C(=O)C(F)(F)F)c2F

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 3/20 0.34
CYP2C9 P11712 1/20 0.34
RORC P51449 4/20 0.33
KEAP1 Q14145 5/20 0.32
NFE2L2 Q16236 5/20 0.32
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
CCNT1 O60563 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CDK9 P50750 1/20 0.31
CCNA1 P78396 1/20 0.31
GYS1 P13807 1/20 0.31
S1PR5 Q9H228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29132485 0.94 CYP2C9 (0.33) PTGER1CYP2C9RORCKMT2AL3MBTL1
SCHEMBL25338437 0.85 NFKB1 (0.36) PTGER1CYP2C9RORCKEAP1NFE2L2
SCHEMBL25339483 0.81 RORC (0.35) PTGER1CYP2C9RORCRXRARXRB
SCHEMBL25338866 0.81 PDE4B (0.33) PTGER1CYP2C9RORCKEAP1NFE2L2
SCHEMBL25340859 0.81 CYP2C9 (0.34) PTGER1CYP2C9RORCKEAP1NFE2L2
SCHEMBL25338244 0.81 KMT2A (0.37) PTGER1CYP2C9RORCKEAP1NFE2L2
SCHEMBL25339196 0.80 RORC (0.35) RORCKEAP1NFE2L2
SCHEMBL29132487 0.80 NFKB1 (0.35) PTGER1CYP2C9RORCKMT2AL3MBTL1
SCHEMBL30683988 0.78 RORC (0.34) PTGER1CYP2C9RORCKMT2AL3MBTL1
SCHEMBL29132483 0.78 RORC (0.34) PTGER1CYP2C9RORCKMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4211122-A1 PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF Calico Life Sciences LLC (US) 2023-07-19 EP disclosed