SCHEMBL25344208

SCHEMBL25344208

CCOC(=O)c1cnn(-c2ccc(F)cc2F)c1NC(=S)NC(=O)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.57
HTT P42858 2/20 0.52
RAB9A P51151 1/20 0.52
GPR35 Q9HC97 2/20 0.48
PAX8 Q06710 1/20 0.47
KDM4E B2RXH2 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
PKM P14618 1/20 0.46
KCNH2 Q12809 1/20 0.46
POLB P06746 3/20 0.44
LMNA P02545 3/20 0.44
MAPT P10636 2/20 0.44
NTRK1 P04629 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ALOX12 P18054 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1355773 0.82 ALDH1A1 (0.59) ALDH1A1HTTRAB9AKDM4ENPSR1
SCHEMBL25342498 0.82 ALDH1A1 (0.49) ALDH1A1HTTRAB9AGPR35PAX8
SCHEMBL22805526 0.80 ALDH1A1 (0.60) ALDH1A1HTTRAB9AKDM4ENPSR1
SCHEMBL1354014 0.80 ALDH1A1 (0.66) ALDH1A1HTTRAB9AKDM4ENPSR1
SCHEMBL1355251 0.79 ALDH1A1 (0.68) ALDH1A1HTTRAB9AKDM4ENPSR1
SCHEMBL174531 0.79 ALDH1A1 (0.59) ALDH1A1HTTRAB9APAX8KDM4E
SCHEMBL24218363 0.79 ALDH1A1 (0.59) ALDH1A1HTTRAB9APAX8KDM4E
SCHEMBL17714338 0.79 PAX8 (0.54) ALDH1A1HTTRAB9APAX8KDM4E
SCHEMBL16252401 0.78 ALDH1A1 (0.48) ALDH1A1HTTRAB9APAX8KDM4E
SCHEMBL5332408 0.75 ALDH1A1 (0.85) ALDH1A1HTTRAB9APAX8KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4472739-A1 IMIDAZOLE MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. Hoffmann-La Roche AG (CH) 2024-12-11 EP disclosed
WO-2023148129-A1 IMIDAZOLE MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2023-08-10 WO disclosed