SCHEMBL25344301

SCHEMBL25344301

Clc1cc(C2COC2)cc(Cl)n1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
S1PR2 O95136 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16210277 0.79 MAP3K12 (0.39)
SCHEMBL31543219 0.79 RAF1 (0.32)
SCHEMBL15535335 0.78 KMT2A (0.37) CYP1A2CYP2D6MAPT
SCHEMBL13738363 0.78 PDE10A (0.34) S1PR2
SCHEMBL15535054 0.77 MAP3K12 (0.46)
SCHEMBL27139379 0.75 RECQL (0.37)
SCHEMBL31224548 0.74 TSHR (0.41) S1PR2
SCHEMBL16216909 0.74 BACE1 (0.34) CYP2D6S1PR2
SCHEMBL16573747 0.73 BACE1 (0.41) CYP2D6MAPT
SCHEMBL31168012 0.73 CHRNB2 (0.43) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4472739-A1 IMIDAZOLE MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. Hoffmann-La Roche AG (CH) 2024-12-11 EP disclosed
WO-2023148129-A1 IMIDAZOLE MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2023-08-10 WO disclosed
CN-114364667-A 3-substituted piperidines for Cbl-b inhibition and the use of Cbl-b inhibitors in combination with cancer vaccines and/or oncolytic viruses 紐力克斯治疗公司 2022-04-15 CN disclosed