SCHEMBL25344387

SCHEMBL25344387

O=C(N1CC2CC(C1)N2)C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 19/20 0.54
CHRNA3 P32297 19/20 0.54
CHRNA4 P43681 19/20 0.54
CHRNB3 Q05901 19/20 0.54
CHRNA6 Q15825 19/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12926722 0.89 CHRNB2 (0.53) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
Trifluoroacetic Acid SCHEMBL993236 0.84 CHRNB2 (0.48) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6
SCHEMBL1711527 0.77 CHRNB2 (0.58) CHRNB2CHRNA3CHRNA4
SCHEMBL1711243 0.77 CHRNB2 (0.58) CHRNB2CHRNA3CHRNA4
SCHEMBL1711255 0.77 CHRNB2 (0.58) CHRNB2CHRNA3CHRNA4
SCHEMBL5387959 0.75 EPHX1 (0.35)
SCHEMBL5387956 0.75 EPHX1 (0.35)
SCHEMBL9235459 0.75 PDK1 (0.36)
SCHEMBL20204150 0.74 GAA (0.42)
SCHEMBL1982249 0.74 CHRNB2 (0.58) CHRNB2CHRNA3CHRNA4CHRNB3CHRNA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4472739-A1 IMIDAZOLE MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. Hoffmann-La Roche AG (CH) 2024-12-11 EP disclosed
WO-2023148129-A1 IMIDAZOLE MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2023-08-10 WO disclosed
WO-2023148129-A1 IMIDAZOLE MACROCYCLES FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2023-08-10 WO disclosed