SCHEMBL25348239

SCHEMBL25348239

COC(=O)c1cc(Br)nc2c1CCC2OC(C)=O

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.36
OPRK1 P41145 12/20 0.34
ALDH1A1 P00352 2/20 0.33
HPGD P15428 1/20 0.33
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
KDM4E B2RXH2 1/20 0.31
S1PR1 P21453 1/20 0.31
ACHE P22303 2/20 0.31
GRIA1 P42261 1/20 0.31
GRIA2 P42262 1/20 0.31
GRIA3 P42263 1/20 0.31
GRIA4 P48058 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30540672 1.00 L3MBTL1 (0.36) L3MBTL1OPRK1ALDH1A1HPGDDDB1
SCHEMBL25348951 0.82 L3MBTL1 (0.39) L3MBTL1OPRK1ALDH1A1HPGDKDM4E
SCHEMBL25348307 0.82 L3MBTL1 (0.39) L3MBTL1OPRK1ALDH1A1HPGD
SCHEMBL22852087 0.70 CHRM4 (0.37)
SCHEMBL25348161 0.69 ACHE (0.51) L3MBTL1ALDH1A1HPGDKDM4EACHE
SCHEMBL8264784 0.68 CYP1A2 (0.35) S1PR1
SCHEMBL25353988 0.68 L3MBTL1 (0.38) L3MBTL1ALDH1A1HPGDKDM4EACHE
SCHEMBL30540629 0.68 L3MBTL1 (0.36) L3MBTL1ALDH1A1HPGDKDM4EACHE
SCHEMBL23976198 0.67 S1PR1 (0.31) S1PR1
SCHEMBL30225223 0.67 S1PR1 (0.31) S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118696043-A Heterocyclic compounds, compositions thereof and methods of treatment therewith 百济神州有限公司 2024-09-24 CN disclosed
WO-2023151642-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE , LTD. (KY) 2023-08-17 WO disclosed
WO-2023151636-A1 HETEROCYCLIC COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH BEIGENE , LTD. (KY) 2023-08-17 WO disclosed