SCHEMBL2536341

SCHEMBL2536341

Cc1ccc(N(C(=O)Nc2ccccc2)c2ncnc(N3CCOCC3)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.50
PIK3CA P42336 4/20 0.48
MTOR P42345 3/20 0.48
PIK3CG P48736 3/20 0.48
HPGD P15428 2/20 0.48
ALDH1A1 P00352 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
LMNA P02545 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KDM4E B2RXH2 1/20 0.44
HIF1A Q16665 1/20 0.44
USP2 O75604 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
BRAF P15056 1/20 0.44
GAA P10253 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
MEN1 O00255 1/20 0.43
ALOX15 P16050 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2536344 0.96 PIK3CA (0.51) PTPN11PIK3CAMTORPIK3CGHPGD
SCHEMBL2535018 0.82 PTPN11 (0.53) PTPN11PIK3CAMTORPIK3CGALDH1A1
SCHEMBL2533509 0.81 PTPN11 (0.53) PTPN11PIK3CAMTORPIK3CGALDH1A1
SCHEMBL2535020 0.81 LMNA (0.47) PTPN11PIK3CAMTORPIK3CGALDH1A1
SCHEMBL2533512 0.81 LMNA (0.45) PTPN11PIK3CAALDH1A1L3MBTL1LMNA
SCHEMBL2535568 0.77 PTPN11 (0.50) PTPN11PIK3CAMTORPIK3CGALDH1A1
SCHEMBL2535576 0.77 PKM (0.41) PTPN11PIK3CAMTORPIK3CGALDH1A1
SCHEMBL29000061 0.76 PIK3CA (0.64) PIK3CAMTORPIK3CGALDH1A1L3MBTL1
SCHEMBL2535323 0.76 PTPN11 (0.49) PTPN11PIK3CAMTORPIK3CGALDH1A1
SCHEMBL2535324 0.76 PIK3CA (0.41) PTPN11PIK3CAMTORPIK3CGALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8039469-B2 Triazine compounds as PI3 kinase and mTOR inhibitors WYETH LLC (US) 2011-10-18 US disclosed