SCHEMBL25378342

SCHEMBL25378342

CCn1cc(Nc2ccccc2)c(C)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.48
LMNA P02545 3/20 0.48
GAA P10253 5/20 0.46
LRRK2 Q5S007 2/20 0.43
CYP1A2 P05177 1/20 0.43
NAMPT P43490 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.40
COMT P21964 1/20 0.40
KDM4E B2RXH2 4/20 0.39
HPGD P15428 4/20 0.39
HTT P42858 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAPT P10636 3/20 0.38
MAPK1 P28482 1/20 0.37
POLB P06746 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CA12 O43570 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25377727 0.77 GAA (0.43) ALDH1A1LMNAGAALRRK2CYP1A2
SCHEMBL31010086 0.77 LRRK2 (0.52) ALDH1A1LMNAGAALRRK2CYP1A2
SCHEMBL31010151 0.71 ALDH1A1 (0.43) ALDH1A1LMNALRRK2CYP1A2NAMPT
SCHEMBL116289 0.65
SCHEMBL12345612 0.65 GAA (0.60) ALDH1A1LMNAGAACYP1A2L3MBTL1
SCHEMBL24977465 0.65 TP53 (0.46) ALDH1A1LMNAGAACYP1A2L3MBTL1
SCHEMBL1803617 0.65 GAA (0.52) ALDH1A1GAACYP1A2KDM4EHPGD
SCHEMBL23115605 0.65 BRD4 (0.49) GAACYP1A2L3MBTL1HTTSMN1; SMN2
Diphenylamine SCHEMBL8204165 0.64 HSD17B10 (0.75) ALDH1A1LMNAGAACYP1A2L3MBTL1
SCHEMBL15131708 0.64 GAA (0.58) ALDH1A1LMNAGAACYP1A2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4482832-A1 5-[7-(3,4-DIHYDRO-1H-ISOQUINOLINE-2-CARBONYL)-1,2,3,4 TETRAHYDROISOQUINOLIN-6-Y L]-1H-PYRROLE-3-CARBOXAMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS PRO-APOPTOTIC AGENTS Les Laboratoires Servier (FR) 2025-01-01 EP disclosed
WO-2023161317-A1 5-[7-(3,4-DIHYDRO-1H-ISOQUINOLINE-2-CARBONYL)-1,2,3,4 TETRAHYDROISOQUINOLIN-6-Y L]-1H-PYRROLE-3-CARBOXAMIDE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS PRO-APOPTOTIC AGENTS LES LABORATOIRES SERVIER (FR) 2023-08-31 WO disclosed