SCHEMBL253921

SCHEMBL253921

C[C@@H](O)[C@@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)C(=O)NO

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.47
CA1 P00915 1/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
PPARG P37231 1/20 0.43
HPGDS O60760 1/20 0.43
ANPEP P15144 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1109169 1.00 CA2 (0.47) CA2CA1NPC1RAB9APPARG
SCHEMBL10272727 1.00 CA2 (0.47) CA2CA1NPC1RAB9APPARG
SCHEMBL1109123 1.00 CA2 (0.47) CA2CA1NPC1RAB9APPARG
SCHEMBL405181 0.93 CA2 (0.49) CA2CA1PPARGHPGDSANPEP
SCHEMBL5450568 0.93 CA2 (0.49) CA2CA1PPARGHPGDSANPEP
SCHEMBL254642 0.89 CA2 (0.47) CA2CA1NPC1RAB9AHPGDS
SCHEMBL1912162 0.89 NPC1 (0.45) NPC1RAB9APPARGHPGDSANPEP
SCHEMBL14400918 0.88
SCHEMBL12837824 0.88
SCHEMBL405336 0.88

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed