SCHEMBL254642

SCHEMBL254642

C[C@@H](O)[C@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)C(=O)NN

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 5/20 0.47
CA1 P00915 3/20 0.47
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
HPGDS O60760 2/20 0.43
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
APEX1 P27695 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP3 P08254 1/20 0.38
MMP7 P09237 1/20 0.38
MMP9 P14780 1/20 0.38
MMP13 P45452 1/20 0.38
ROCK2 O75116 1/20 0.38
RPS6KA5 O75582 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1109123 0.89 CA2 (0.47) CA2CA1NPC1RAB9AHPGDS
SCHEMBL253921 0.89 CA2 (0.47) CA2CA1NPC1RAB9AHPGDS
SCHEMBL10272727 0.89 CA2 (0.47) CA2CA1NPC1RAB9AHPGDS
SCHEMBL1912134 0.89 NPC1 (0.52) CA2CA1NPC1RAB9AHPGDS
SCHEMBL1109169 0.89 CA2 (0.47) CA2CA1NPC1RAB9AHPGDS
SCHEMBL19262702 0.88 CA2 (0.44) CA2CA1NPC1RAB9A
SCHEMBL157589 0.85 CA2 (0.42) CA2CA1NPC1RAB9A
SCHEMBL254371 0.85 CA2 (0.42) CA2CA1NPC1RAB9A
SCHEMBL254283 0.85 CA2 (0.63) CA2CA1NPC1RAB9AHPGDS
SCHEMBL254637 0.85 CA2 (0.63) CA2CA1NPC1RAB9AHPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed