SCHEMBL254229

SCHEMBL254229

COC(=O)c1ccc(C#Cc2ccc(N)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.59
APP P05067 3/20 0.53
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
CA12 O43570 1/20 0.52
CA7 P43166 1/20 0.52
CA9 Q16790 1/20 0.52
CA14 Q9ULX7 1/20 0.52
MAPT P10636 4/20 0.52
GAA P10253 2/20 0.50
LOXL2 Q9Y4K0 1/20 0.50
MAPK1 P28482 1/20 0.50
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
MAOA P21397 1/20 0.50
TSHR P16473 1/20 0.48
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3019329 0.93 PTPN11 (0.53) PTPN11APPCA1CA2TDP1
SCHEMBL69268 0.90 PTPN11 (0.69) PTPN11CA1CA2TDP1CA12
SCHEMBL1535874 0.89 PTPN11 (0.63) PTPN11CA1CA2TDP1CA12
SCHEMBL42732 0.88 CA1 (0.64) CA1CA2TDP1CA12CA7
Hydrochloric Acid SCHEMBL8359634 0.86 CA1 (0.61) CA1CA2TDP1CA12CA7
SCHEMBL28108955 0.86 CA1 (0.61) CA1CA2TDP1CA12CA7
SCHEMBL8272575 0.85 PTPN11 (0.58) PTPN11CA1CA2TDP1CA12
SCHEMBL15235703 0.83 MAPT (0.54) PTPN11APPCA1CA2TDP1
SCHEMBL15235704 0.83 MAPT (0.54) PTPN11APPCA1CA2TDP1
SCHEMBL16140276 0.83 TDP1 (0.77) PTPN11CA1CA2TDP1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3448375-B1 BENZOYLGLYCINE DERIVATIVES AND METHODS OF MAKING AND USING SAME UNIV DUKE (US) 2023-09-27 EP disclosed
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed