SCHEMBL25428296

SCHEMBL25428296

CN(C)C(=O)C1CCCN1c1ccc2[nH]cnc2c1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SYK P43405 3/20 0.42
PIK3CA P42336 1/20 0.41
ALDH1A1 P00352 2/20 0.40
HPGD P15428 1/20 0.40
PIK3C3 Q8NEB9 1/20 0.40
CDK2 P24941 1/20 0.39
HSD11B1 P28845 9/20 0.38
CASP3 P42574 1/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31150480 1.00 SYK (0.42) SYKPIK3CAALDH1A1HPGDPIK3C3
SCHEMBL25949040 0.75 ALDH1A1 (0.36) PIK3CAALDH1A1HPGDHSD11B1KDM4E
SCHEMBL31150453 0.72 AR (0.37) PIK3CAALDH1A1HPGDHSD11B1KDM4E
SCHEMBL25425906 0.72 AR (0.37) PIK3CAALDH1A1HPGDHSD11B1KDM4E
SCHEMBL13724767 0.72 SYK (0.49) SYKALDH1A1PIK3C3CDK2CASP3
SCHEMBL3550347 0.72 SYK (0.49) SYKALDH1A1PIK3C3CDK2CASP3
SCHEMBL1673469 0.71 NUDT1 (0.46) PIK3C3
SCHEMBL1444384 0.70 QPCT (0.42) ALDH1A1HPGDKDM4EMAPT
SCHEMBL1444563 0.70 NR3C2 (0.49)
SCHEMBL1445163 0.70 DYRK1A (0.43) ALDH1A1HSD11B1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4466258-A1 NEW BENZIMIDAZOLE PYRIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2024-11-27 EP disclosed
WO-2023139085-A1 NEW BENZIMIDAZOLE PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2023-07-27 WO disclosed
WO-2023139085-A1 NEW BENZIMIDAZOLE PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2023-07-27 WO disclosed