SCHEMBL25435331

SCHEMBL25435331

CN(CCc1ccccc1)S(=O)(=O)c1cc(F)c(O)c2ncccc12

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
COMT P21964 9/20 0.54
HSD17B10 Q99714 1/20 0.47
ALDH1A1 P00352 2/20 0.46
HPGD P15428 1/20 0.46
KDM4E B2RXH2 4/20 0.42
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17962333 0.83 KDM4E (0.58) COMTALDH1A1HPGDKDM4EKMT2A
SCHEMBL17962316 0.78 COMT (0.56) COMTALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL25408540 0.78 COMT (0.56) COMTALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL7684587 0.72 KDM4E (0.64) COMTALDH1A1HPGDKDM4EMAPT
SCHEMBL17960016 0.72 COMT (0.69) COMTALDH1A1HPGDKDM4EMAPT
SCHEMBL17962266 0.71 ALDH1A1 (0.62) COMTALDH1A1HPGDKDM4EKMT2A
SCHEMBL17962325 0.70 COMT (1.00) COMTALDH1A1KDM4ESMN1; SMN2TDP1
SCHEMBL17960013 0.69 COMT (1.00) COMTALDH1A1KDM4EMAPTTDP1
SCHEMBL7689814 0.68 COMT (0.57) COMTALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL17962259 0.68 KDM4E (0.63) COMTHSD17B10ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3250209-B1 COMT INHIBITING METHODS AND COMPOSITIONS LIEBER INST FOR BRAIN DEVELOPMENT (US) 2023-09-13 EP claimed