SCHEMBL25436239

SCHEMBL25436239

O=C(O)c1cnc(Cl)nc1NCc1cccc(F)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM5A P29375 1/20 0.51
KDM4C Q9H3R0 1/20 0.51
KDM5B Q9UGL1 1/20 0.51
NTRK1 P04629 8/20 0.51
RPS6KB1 P23443 3/20 0.48
AURKA O14965 2/20 0.48
AURKB Q96GD4 1/20 0.48
JAK2 O60674 1/20 0.48
JAK1 P23458 1/20 0.48
JAK3 P52333 1/20 0.48
CCNT1 O60563 2/20 0.48
STAT6 P42226 1/20 0.46
APP P05067 1/20 0.46
ADORA3 P0DMS8 1/20 0.45
FFAR1 O14842 1/20 0.44
ADORA2A P29274 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22261068 0.89 JAK2 (0.59) NTRK1RPS6KB1AURKAAURKBJAK2
SCHEMBL4188524 0.88 CSNK2A2 (0.51) KDM5AKDM4CKDM5BRPS6KB1JAK3
Hydrochloric Acid SCHEMBL4178767 0.87 CSNK2A2 (0.50) KDM5AKDM4CKDM5BRPS6KB1JAK3
SCHEMBL25435346 0.85 P4HTM (0.51) RPS6KB1AURKAJAK3STAT6ADORA3
SCHEMBL28713125 0.83 NTRK1 (0.62) NTRK1CCNT1
SCHEMBL29392704 0.83 NTRK1 (0.62) NTRK1CCNT1
SCHEMBL25435320 0.83 VNN1 (0.54) JAK2JAK3
SCHEMBL15584955 0.80 NTRK1 (0.50) NTRK1AURKAAURKBJAK2JAK3
SCHEMBL19675773 0.80 NTRK1 (0.51) NTRK1AURKAAURKBJAK2JAK3
SCHEMBL29608147 0.80 NTRK1 (0.51) NTRK1AURKAAURKBJAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3686197-B1 2-SUBSTITUTED PYRAZOLE AMINO-4-SUBSTITUTED AMINO-5-PYRIMIDINE FORMAMIDE COMPOUND, COMPOSITION, AND APPLICATION THEREOF BEIJING SCITECH MQ PHARMACEUTICALS LTD (CN) 2023-06-21 EP disclosed