SCHEMBL25436735

SCHEMBL25436735

CS(=O)(=O)c1ccc(S(=O)(=O)N2CCC3(CC2)CNc2ccccc23)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OXTR P30559 1/20 0.44
TSHR P16473 1/20 0.43
ALDH1A1 P00352 3/20 0.41
KMT2A Q03164 2/20 0.41
CYP2D6 P10635 1/20 0.41
MEN1 O00255 1/20 0.41
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TNKS O95271 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
CYP2C19 P33261 2/20 0.40
POLB P06746 1/20 0.40
CCR5 P51681 1/20 0.40
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
USP2 O75604 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5578474 0.88 SMN1; SMN2 (0.51) ALDH1A1KMT2AMEN1L3MBTL1POLB
SCHEMBL30413328 0.84 CYP3A4 (0.40) OXTRTSHRALDH1A1KMT2ACYP2D6
SCHEMBL38333 0.84 CYP2C9 (0.46) TSHRALDH1A1KMT2ACYP2D6MEN1
Hydrochloric Acid SCHEMBL7012082 0.83 CYP2C9 (0.44) TSHRALDH1A1KMT2ACYP2D6MEN1
SCHEMBL7013380 0.80 TNKS (0.46) ALDH1A1KMT2ACYP2D6MEN1MAPK1
Hydrochloric Acid SCHEMBL7006808 0.79 TNKS (0.43) ALDH1A1TNKSTNKS2POLBCCR5
Hydrochloric Acid SCHEMBL7006198 0.79 TNKS (0.45) ALDH1A1KMT2ACYP2D6MEN1MAPK1
SCHEMBL30412930 0.73 TSHR (0.51) TSHRALDH1A1KMT2ATNKSTNKS2
SCHEMBL1670650 0.73 TNKS (0.46) TNKSTNKS2CCR5
Hydrochloric Acid SCHEMBL25230408 0.72 TNKS (0.45) TNKSTNKS2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4192957-A2 TRPML MODULATORS Casma Therapeutics, Inc. (US) 2023-06-14 EP disclosed
WO-2022032073-A2 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2022-02-10 WO disclosed