SCHEMBL7013380

SCHEMBL7013380

NS(=O)(=O)N1CCC2(CC1)CNc1ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 2/20 0.46
TNKS2 Q9H2K2 2/20 0.46
AVPR1A P37288 1/20 0.43
KCNH2 Q12809 2/20 0.43
HDAC1 Q13547 2/20 0.43
CCR5 P51681 1/20 0.40
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
OPRD1 P41143 1/20 0.36
KDM1A O60341 1/20 0.36
PRNP P04156 1/20 0.35
CHRNA7 P36544 3/20 0.35
NPY5R Q15761 2/20 0.33
CYP2D6 P10635 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
BACE1 P56817 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7006198 0.98 TNKS (0.45) TNKSTNKS2AVPR1AKCNH2HDAC1
SCHEMBL38333 0.87 CYP2C9 (0.46) TNKSTNKS2AVPR1AKCNH2HDAC1
Hydrochloric Acid SCHEMBL7012082 0.85 CYP2C9 (0.44) TNKSTNKS2AVPR1AKCNH2HDAC1
Hydrochloric Acid SCHEMBL7006808 0.84 TNKS (0.43) TNKSTNKS2AVPR1AKCNH2HDAC1
SCHEMBL30412930 0.81 TSHR (0.51) TNKSTNKS2ALDH1A1KMT2A
SCHEMBL15007673 0.81 TNKS (0.46) TNKSTNKS2AVPR1AKCNH2HDAC1
SCHEMBL25436735 0.80 OXTR (0.44) TNKSTNKS2CCR5CYP2D6MEN1
SCHEMBL5578474 0.80 SMN1; SMN2 (0.51) AVPR1ACCR5MEN1ALDH1A1KMT2A
SCHEMBL14624333 0.78 TNKS (0.47) TNKSTNKS2AVPR1AKCNH2HDAC1
SCHEMBL29479467 0.78 TNKS (0.44) TNKSTNKS2AVPR1AKCNH2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1129089-A4 SPIRO-INDOLINES AS Y5 RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2003-01-22 EP disclosed
EP-1129089-A1 SPIRO-INDOLINES AS Y5 RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2001-09-05 EP disclosed
WO-2000027845-A1 SPIRO-INDOLINES AS Y5 RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-05-18 WO disclosed