SCHEMBL254523

SCHEMBL254523

CCCCCCCCC=CCCCCCCCCN(CCCCCCCCC=CCCCCCCCC)CC(O)CO

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGKA P23743 1/20 0.49
SPHK2 Q9NRA0 4/20 0.46
SPHK1 Q9NYA1 4/20 0.46
CETP P11597 3/20 0.46
MEN1 O00255 3/20 0.45
MAPT P10636 3/20 0.45
KMT2A Q03164 3/20 0.45
ALDH1A1 P00352 3/20 0.45
GMNN O75496 2/20 0.45
LMNA P02545 2/20 0.45
GLA P06280 2/20 0.45
POLB P06746 2/20 0.45
THRB P10828 2/20 0.45
MAPK1 P28482 2/20 0.45
CXCR5 P32302 2/20 0.45
CCR6 P51684 2/20 0.45
BLM P54132 2/20 0.45
UBE2N P61088 2/20 0.45
CYP2D6 P10635 2/20 0.45
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL254521 1.00 DGKA (0.49) DGKASPHK2SPHK1CETPMEN1
SCHEMBL12735352 0.95 FAAH (0.50) DGKAALDH1A1LMNAALOX15FAAH
SCHEMBL30469 0.95 FAAH (0.50) DGKAALDH1A1LMNAALOX15FAAH
SCHEMBL16694673 0.95 FAAH (0.50) DGKAALDH1A1LMNAALOX15FAAH
SCHEMBL12664404 0.95 FAAH (0.50) DGKAALDH1A1LMNAALOX15FAAH
SCHEMBL1288253 0.89 USP2 (0.46) SPHK1CETPMEN1MAPTKMT2A
SCHEMBL3673713 0.89 USP2 (0.46) SPHK1CETPMEN1MAPTKMT2A
SCHEMBL11405257 0.89 USP2 (0.46) SPHK1CETPMEN1MAPTKMT2A
SCHEMBL1288234 0.89 USP2 (0.46) SPHK1CETPMEN1MAPTKMT2A
SCHEMBL3669886 0.89 USP2 (0.46) SPHK1CETPMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 509 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022115739-A1 2022-06-02 WO claimed
EP-4735033-A2 MRNA-ENCODED TAT WITH ATTENUATED CYTOTOXICITY FOR HIV AND SIV LATENCY REVERSAL The Trustees of the University of Pennsylvania (US) 2026-05-06 EP disclosed
WO-2025128913-A1 INHIBITION OF ENDOSOMAL ESCAPE DETECTION TO AMELIORATE THE INFLAMMATORY SIDE-EFFECTS OF LIPID NANOPARTICLES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2025-06-19 WO disclosed
WO-2025129106-A1 IMMUNOEVASIVE TARGETING MOLECULES FOR EFFICIENT TARGETED DELIVERY THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2025-06-19 WO disclosed
WO-2025111442-A1 LIPID NANOPARTICLES AND METHODS OF USE FOR DNA DELIVERY THE WISTAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2025-05-30 WO disclosed
WO-2025080672-A1 IMMUNE CELL TARGETED DELIVERY VEHICLES AND METHODS OF USE THEREOF THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2025-04-17 WO disclosed
EP-4531905-A1 RNA COMPOSITIONS FOR DELIVERY OF MONKEYPOX ANTIGENS AND RELATED METHODS BioNTech SE (DE) 2025-04-09 EP disclosed
WO-2025072623-A1 COMPOSITIONS AND METHODS FOR TARGETING IMMUNE CELLS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2025-04-03 WO disclosed
WO-2025038627-A2 PENTAERYTHRITOL-BASED IONIZABLE AMPHIPHILIC JANUS DENDRIMERS, DELIVERY SYSTEMS COMPRISING THEREOF, AND METHODS OF USE THEREOF THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2025-02-20 WO disclosed
WO-2025030103-A1 RNA COMPOSITIONS ENCODING HERPES SIMPLEX VIRUS GLYCOPROTEIN B ANTIGENS AND USES THEREOF THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2025-02-06 WO disclosed
WO-2011000107-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS TO SOLID TUMORS PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-01-06 WO disclosed
EP-2224912-A1 IMPROVED COMPOSITIONS AND METHODS FOR THE DELIVERY OF NUCLEIC ACIDS TEKMIRA Pharmaceuticals Corporation (CA) 2010-09-08 EP disclosed
WO-2010083615-A1 COMPOSITIONS AND METHODS FOR SILENCING APOLIPOPROTEIN C-III EXPRESSION PROTIVA BIOTHERAPEUTICS, INC. (CA) 2010-07-29 WO disclosed
WO-2010068816-A1 GNAQ TARGETED DSRNA COMPOSITIONS AND METHODS FOR INHIBITING EXPRESSION ALNYLAM PHARMACEUTICALS, INC. (US) 2010-06-17 WO disclosed
US-20100130588-A1 NOVEL LIPID FORMULATIONS FOR NUCLEIC ACID DELIVERY PROTIVA BIOTHERAPEUTICS, INC. (CA) 2010-05-27 US disclosed
WO-2009132131-A1 AMINO LIPID BASED IMPROVED LIPID FORMULATION ALNYLAM PHARMACEUTICALS, INC. (US) 2009-10-29 WO disclosed
WO-2009129319-A2 SILENCING OF CSN5 GENE EXPRESSION USING INTERFERING RNA PROTIVA BIOTHERAPEUTICS, INC. (CA) 2009-10-22 WO disclosed
WO-2009127060-A1 NOVEL LIPID FORMULATIONS FOR NUCLEIC ACID DELIVERY PROTIVA BIOTHERAPEUTICS, INC. (CA) 2009-10-22 WO disclosed
WO-2009088891-A1 SCREENING METHOD FOR SELECTED AMINO LIPID-CONTAINING COMPOSITIONS ALNYLAM PHARMACEUTICALS, INC. (US) 2009-07-16 WO disclosed
WO-2009086558-A1 IMPROVED COMPOSITIONS AND METHODS FOR THE DELIVERY OF NUCLEIC ACIDS TEKMIRA PHARMACEUTICALS CORPORATION (CA) 2009-07-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100130588-A1 NOVEL LIPID FORMULATIONS FOR NUCLEIC ACID DELIVERY SARNP, NPC1L1, SNRPE DGKA 1204/4885SPHK2 177/4885SPHK1 192/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.