SCHEMBL2545345

SCHEMBL2545345

CC(CNC(=O)O)c1ccc(Br)cc1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 1/20 0.41
APLNR P35414 4/20 0.41
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40
MMP7 P09237 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40
CYP3A4 P08684 1/20 0.40
PTGFR P43088 1/20 0.40
ACACB O00763 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ALDH1A1 P00352 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
DGAT1 O75907 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15092576 0.81 AAK1 (0.53) APLNR
SCHEMBL29784722 0.81 AAK1 (0.53) APLNR
SCHEMBL15092577 0.81 AAK1 (0.53) APLNR
SCHEMBL8243599 0.80 APLNR (0.43) FPR2APLNRMMP1MMP2MMP3
SCHEMBL27008783 0.77 FPR2 (0.44) FPR2APLNRMMP1MMP2MMP3
SCHEMBL15092388 0.77 FPR2 (0.44) FPR2APLNRMMP1MMP2MMP3
SCHEMBL15092400 0.76 APLNR (0.44) FPR2APLNRMMP1MMP2MMP3
SCHEMBL12267174 0.76 APLNR (0.44) FPR2APLNRMMP1MMP2MMP3
SCHEMBL2879129 0.76 APLNR (0.44) FPR2APLNRMMP1MMP2MMP3
SCHEMBL14274718 0.75 APLNR (0.44) FPR2APLNRMMP1MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2552206-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-02-06 EP disclosed
WO-2011123419-A1 TRYCYCLIC COMPOUNDS AND PBK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2011-10-06 WO disclosed