SCHEMBL254722

SCHEMBL254722

C[C@@H](O)[C@H](NC(=O)c1ccc(OCc2ccc(N)cc2)cc1)C(=O)NO

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.52
ALDH1A1 P00352 3/20 0.49
MAPT P10636 3/20 0.49
MAPK1 P28482 1/20 0.49
HTT P42858 1/20 0.49
PSMB1 P20618 1/20 0.47
PSMB8 P28062 1/20 0.47
PSMB9 P28065 1/20 0.47
PSMB5 P28074 1/20 0.47
PSMB10 P40306 1/20 0.47
PSMB2 P49721 1/20 0.47
RXRA P19793 1/20 0.46
RXRB P28702 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
PARP10 Q53GL7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL254370 1.00 PPARG (0.52) PPARGALDH1A1MAPTMAPK1HTT
SCHEMBL254798 0.87 MAPT (0.53) PPARGALDH1A1MAPTMAPK1HTT
SCHEMBL402664 0.86 PPARG (0.49) PPARGPSMB1PSMB8PSMB9PSMB5
SCHEMBL156853 0.83 ADAM17 (0.51) PPARG
SCHEMBL15235701 0.83 ADAM17 (0.51) PPARG
SCHEMBL15235707 0.83 ADAM17 (0.51) PPARG
SCHEMBL15227935 0.83 ADAM17 (0.51) PPARG
SCHEMBL10272727 0.81 CA2 (0.47) PPARG
SCHEMBL1109123 0.81 CA2 (0.47) PPARG
SCHEMBL1109169 0.81 CA2 (0.47) PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed