SCHEMBL254965

SCHEMBL254965

O=C(Nc1c(F)c(F)c(F)c(F)c1F)c1ccc(-c2ccc(CO)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.47
NAMPT P43490 1/20 0.44
TSHR P16473 2/20 0.43
NR1H4 Q96RI1 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
F2 P00734 1/20 0.43
PLG P00747 1/20 0.43
PLAU P00749 1/20 0.43
PLAT P00750 1/20 0.43
KLKB1 P03952 1/20 0.43
PRSS1 P07477 1/20 0.43
HDAC6 Q9UBN7 3/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC3 O15379 2/20 0.41
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15235770 0.84 NAMPT (0.40) NAMPTTSHRNPSR1LMNAMEN1
SCHEMBL14716260 0.82 TSHR (0.56) PTPN1TSHRNPSR1LMNAMEN1
SCHEMBL18837905 0.74 PLK1 (0.63) TSHRNR1H4HDAC6EPHX2HDAC8
SCHEMBL4586310 0.73 TSHR (0.60) PTPN1TSHRNPSR1LMNAMEN1
SCHEMBL2915005 0.70 TSHR (0.56) TSHRNPSR1LMNAMEN1KMT2A
SCHEMBL2642122 0.69 PTPN1 (0.67) PTPN1NAMPTNR1H4MEN1KMT2A
SCHEMBL3641834 0.69 RARB (0.58) TSHRNR1H4MEN1KMT2AEPHX2
SCHEMBL20424311 0.69 HDAC6 (0.67) HDAC6HDAC1HDAC3HDAC8HDAC2
SCHEMBL1364607 0.69 MPO (0.61) LMNAPRSS1HDAC6HDAC3EPHX2
SCHEMBL12440876 0.68 NR1H4 (0.62) PTPN1NR1H4LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed