SCHEMBL255108

SCHEMBL255108

C[C@](O)(c1ccc(O)cc1)[C@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)C(=O)NO

nearest known ligand 0.78

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 1/20 0.43
ESRRG P62508 2/20 0.38
EPHX2 P34913 1/20 0.37
HDAC1 Q13547 1/20 0.37
ESRRB O95718 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19262704 0.90 APP (0.42)
SCHEMBL19262705 0.90 APP (0.42)
SCHEMBL15235682 0.88
SCHEMBL15235689 0.88
SCHEMBL15235774 0.88
SCHEMBL15235773 0.88
SCHEMBL158012 0.88
SCHEMBL255220 0.85 NPC1 (0.41) ESRRGNPC1RAB9A
SCHEMBL10272722 0.83 NPC1 (0.42) ESRRGEPHX2HDAC1ESRRBNPC1
SCHEMBL13984823 0.82 ANPEP (0.48) ANPEPHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed