SCHEMBL255220

SCHEMBL255220

CC(C)(O)[C@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)C(=O)NO

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
CA2 P00918 1/20 0.40
ESRRG P62508 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13267172 0.89 NPC1 (0.41) NPC1RAB9ACA2ESRRG
SCHEMBL10287224 0.87 HPGDS (0.51) NPC1RAB9A
SCHEMBL254900 0.87 ANPEP (0.39) NPC1RAB9A
SCHEMBL13266885 0.86 ANPEP (0.52) NPC1
SCHEMBL13245022 0.86
SCHEMBL254610 0.86 ANPEP (0.41) NPC1RAB9AESRRG
SCHEMBL405554 0.85 TAS1R3 (0.50) NPC1RAB9A
SCHEMBL255108 0.85 ANPEP (0.43) NPC1RAB9AESRRG
SCHEMBL13459333 0.84 NPC1 (0.43) NPC1RAB9ACA2ESRRG
SCHEMBL13266884 0.84 EPHX2 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed
US-20100190766-A1 ANTIBACTERIAL AGENTS ACHAOGEN, INC. (US) 2010-07-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100190766-A1 ANTIBACTERIAL AGENTS MRPL21, SI, ABCB11 NPC1 299/4885RAB9A 509/4885CA2 3489/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.