SCHEMBL10272722

SCHEMBL10272722

C[C@@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)[C@](C)(O)c1ccc(O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
HPGDS O60760 2/20 0.41
EPHX2 P34913 1/20 0.40
ESRRG P62508 4/20 0.39
HSD17B1 P14061 1/20 0.38
MPO P05164 1/20 0.38
CYP3A4 P08684 1/20 0.38
KDM5A P29375 1/20 0.38
BLM P54132 1/20 0.38
GFER P55789 1/20 0.38
PMP22 Q01453 1/20 0.38
HIF1A Q16665 1/20 0.38
HDAC1 Q13547 1/20 0.38
DEGS1 O15121 1/20 0.38
NR1H4 Q96RI1 1/20 0.37
PTGS1 P23219 2/20 0.37
ESRRB O95718 1/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL255108 0.83 ANPEP (0.43) NPC1RAB9AEPHX2ESRRGHDAC1
SCHEMBL10272711 0.77 HPGDS (0.34) NPC1RAB9AHPGDSEPHX2ESRRG
SCHEMBL19262704 0.72 APP (0.42)
SCHEMBL19262705 0.72 APP (0.42)
SCHEMBL15235682 0.71
SCHEMBL15235773 0.71
SCHEMBL254376 0.70 CA2 (0.43) NPC1RAB9AHPGDSEPHX2ESRRG
SCHEMBL255220 0.70 NPC1 (0.41) NPC1RAB9AESRRG
SCHEMBL853579 0.69 MLYCD (0.59) NPC1RAB9ACYP3A4HIF1AMEN1
Bisphenol A SCHEMBL28319737 0.69 ESR1 (0.67) ESRRGCYP3A4HIF1ALMNATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed