SCHEMBL25519368

SCHEMBL25519368

CCN1CCC[C@@H](Nc2cc(C)c(Cl)nn2)C1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 13/20 0.57
IL1B P01584 7/20 0.52
KCNH2 Q12809 1/20 0.52
CAMK2D Q13557 2/20 0.48
ADORA2A P29274 1/20 0.46
TNF P01375 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30517832 1.00 NLRP3 (0.57) NLRP3IL1BKCNH2CAMK2DADORA2A
SCHEMBL25303253 0.87 NLRP3 (0.55) NLRP3IL1BKCNH2TNF
SCHEMBL25254731 0.87 NLRP3 (0.55) NLRP3IL1BKCNH2TNF
SCHEMBL29270330 0.86 NLRP3 (0.57) NLRP3IL1BKCNH2CAMK2DADORA2A
SCHEMBL25300069 0.86 NLRP3 (0.51) NLRP3IL1BKCNH2CAMK2DTNF
SCHEMBL25300070 0.86 NLRP3 (0.51) NLRP3IL1BKCNH2CAMK2DTNF
SCHEMBL31021469 0.85 NLRP3 (0.48) NLRP3IL1BKCNH2CAMK2DADORA2A
SCHEMBL31367803 0.85 NLRP3 (0.57) NLRP3IL1BKCNH2CAMK2DADORA2A
SCHEMBL29030489 0.85 IL1B (0.48) NLRP3IL1BKCNH2TNF
SCHEMBL25304051 0.85 IL1B (0.48) NLRP3IL1BKCNH2TNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118265701-A Pyridazine derivatives as inhibitors of NLRP3 豪夫迈·罗氏有限公司 2024-06-28 CN disclosed
WO-2023088987-A1 PYRIDAZINE DERIVATIVES AS INHIBITORS OF NLRP3 F. HOFFMANN-LA ROCHE AG (CH) 2023-05-25 WO disclosed