SCHEMBL25522892

SCHEMBL25522892

CCCNc1c(N(C)C)c(=O)c1=O

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.34
ALDH1A1 P00352 2/20 0.34
GAA P10253 2/20 0.33
ADAMTS5 Q9UNA0 1/20 0.33
MCL1 Q07820 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 2/20 0.32
LMNA P02545 2/20 0.32
BACH1 O14867 1/20 0.32
MAFK O60675 1/20 0.32
GRIN2D O15399 2/20 0.32
GRIN3B O60391 2/20 0.32
GRIN1 Q05586 2/20 0.32
GRIN2A Q12879 2/20 0.32
GRIN2B Q13224 2/20 0.32
GRIN2C Q14957 2/20 0.32
GRIN3A Q8TCU5 2/20 0.32
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22645978 0.84 ADAMTS5 (0.35) MAPTALDH1A1GAAADAMTS5MCL1
SCHEMBL22645840 0.82 GAA (0.31) GAA
SCHEMBL21231164 0.82 GAA (0.31) GAA
SCHEMBL23783545 0.82 GRIN2D (0.32) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL21842751 0.82 MCL1 (0.34) MAPTALDH1A1GAAMCL1L3MBTL1
SCHEMBL24263719 0.81 ALDH1A1 (0.42) MAPTALDH1A1ADAMTS5
SCHEMBL24968964 0.79 ALDH1A1 (0.41) ALDH1A1
SCHEMBL13918748 0.79 GAA (0.41) MAPTALDH1A1GAAKDM4ELMNA
SCHEMBL21473465 0.79
SCHEMBL22645938 0.79 CYP1A2 (0.38) ALDH1A1GAAL3MBTL1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230150946-A1 HETEROCYCLE CONTAINING STAT INHIBITORS AND COMPOSITIONS OXFORD FINANCE LLC 2023-05-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230150946-A1 HETEROCYCLE CONTAINING STAT INHIBITORS AND COMPOSITIONS STAT5A, STAT5B, STAT3 MAPT 4617/4885ALDH1A1 4293/4885GAA 2500/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.