SCHEMBL25523969

SCHEMBL25523969

CN1Cc2cc(N)ncc2C1=O

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 4/20 0.40
GABRA1 P14867 1/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
PRF1 P14222 12/20 0.36
MKNK1 Q9BUB5 1/20 0.36
ALK Q9UM73 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21403857 0.79 LRRK2 (0.45) LRRK2GABRA1PRF1MKNK1
SCHEMBL30397487 0.79 LRRK2 (0.45) LRRK2GABRA1PRF1MKNK1
SCHEMBL29084843 0.79 LRRK2 (0.40) LRRK2GABRA1PRF1MKNK1
SCHEMBL25289133 0.79 LRRK2 (0.40) LRRK2GABRA1PRF1MKNK1
SCHEMBL25421259 0.79 LRRK2 (0.40) LRRK2GABRA1PRF1MKNK1
SCHEMBL15571453 0.77 PRF1 (0.46) PRF1
SCHEMBL29084811 0.77 GABRA1 (0.47) LRRK2GABRA1PRF1MKNK1
SCHEMBL25512529 0.77 LRRK2 (0.38) LRRK2GABRA1PRF1MKNK1
SCHEMBL23349324 0.74 GABRA1 (0.39) LRRK2GABRA1MKNK1
SCHEMBL15571500 0.74 PRF1 (0.56) PRF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed