SCHEMBL25524262

SCHEMBL25524262

CC(=N)C(=O)c1ccnc(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
IDO1 P14902 1/20 0.37
AR P10275 4/20 0.35
KDM4C Q9H3R0 4/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM5C P41229 3/20 0.35
CA12 O43570 2/20 0.35
CA9 Q16790 2/20 0.35
KDM6B O15054 2/20 0.35
KDM2A Q9Y2K7 2/20 0.35
KDM3A Q9Y4C1 2/20 0.35
KDM4A O75164 2/20 0.35
KDM5B Q9UGL1 2/20 0.35
TET3 O43151 1/20 0.35
BBOX1 O75936 1/20 0.35
MAPT P10636 1/20 0.35
KDM5A P29375 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL220172 0.81 KDM1A (0.44) KDM1AHDAC1HDAC6IDO1AR
SCHEMBL30595888 0.81 KDM1A (0.44) KDM1AHDAC1HDAC6IDO1AR
SCHEMBL3466541 0.81 IDO1 (0.41) KDM1AHDAC1HDAC6IDO1AR
Bromide SCHEMBL6203968 0.79 KDM1A (0.42) KDM1AHDAC1HDAC6IDO1AR
SCHEMBL25263407 0.79 KDM1A (0.42) KDM1AHDAC1HDAC6IDO1AR
SCHEMBL28786825 0.77 LMNA (0.47) KDM1AHDAC1HDAC6IDO1AR
SCHEMBL3465859 0.77 IDO1 (0.39) KDM1AHDAC1HDAC6IDO1AR
SCHEMBL3124147 0.75 KDM1A (0.40) KDM1AHDAC1HDAC6IDO1AR
SCHEMBL40395 0.75 KDM4C (0.61) KDM1AHDAC1HDAC6KDM4CKDM4E
SCHEMBL30527973 0.75 KDM4C (0.61) KDM1AHDAC1HDAC6KDM4CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed