SCHEMBL25525166

SCHEMBL25525166

N[C@@H]1CCC[C@H](c2nnc3c(Cl)nccn23)C1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 11/20 0.37
ADORA3 P0DMS8 4/20 0.35
NR1I2 O75469 1/20 0.35
BTK Q06187 1/20 0.33
TNK2 Q07912 1/20 0.33
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32
PTPN11 Q06124 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30396230 1.00 HSD11B1 (0.37) HSD11B1ADORA3NR1I2BTKTNK2
SCHEMBL21138249 0.87 HSD11B1 (0.45) HSD11B1ADORA3NR1I2TNK2CCNE1
SCHEMBL21138331 0.86 HSD11B1 (0.47) HSD11B1ADORA3NR1I2CCNE1CDK2
SCHEMBL25525429 0.85 HSD11B1 (0.34) HSD11B1ADORA3NR1I2BTKTNK2
SCHEMBL21138816 0.84 HSD11B1 (0.49) HSD11B1ADORA3NR1I2CCNE1CDK2
SCHEMBL21057446 0.84 HSD11B1 (0.37) HSD11B1ADORA3NR1I2CCNE1CDK2
SCHEMBL19917049 0.84 HSD11B1 (0.37) HSD11B1ADORA3NR1I2CCNE1CDK2
SCHEMBL21138374 0.81 HSD11B1 (0.35) HSD11B1ADORA3NR1I2TNK2
SCHEMBL21159124 0.80 HSD11B1 (0.37) HSD11B1ADORA3NR1I2CCNE1CDK2
SCHEMBL21159625 0.80 HSD11B1 (0.33) HSD11B1ADORA3NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed