SCHEMBL255253

SCHEMBL255253

Nc1ccc(-c2ccc(C(=O)N[C@H](C(=O)NO)[C@H](O)c3ccc(O)cc3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 11/20 0.50
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
HPGDS O60760 1/20 0.39
HDAC1 Q13547 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19262601 0.89 APP (0.44)
SCHEMBL19262698 0.89 APP (0.44)
SCHEMBL254675 0.87 APP (0.39) ANPEP
SCHEMBL15235772 0.87 APP (0.39) ANPEP
SCHEMBL15235688 0.87 APP (0.39) ANPEP
SCHEMBL157159 0.87 APP (0.39) ANPEP
SCHEMBL10272727 0.80 CA2 (0.47) ANPEPCA1CA2HPGDS
SCHEMBL1109169 0.80 CA2 (0.47) ANPEPCA1CA2HPGDS
SCHEMBL1109123 0.80 CA2 (0.47) ANPEPCA1CA2HPGDS
SCHEMBL403655 0.80 HPGDS (0.59) ANPEPCA1CA2HPGDSHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed