SCHEMBL25528340

SCHEMBL25528340

C[C@@H]1C(=O)N(C)c2cc(-c3ccc4[nH]ncc4c3)ccc2C(=O)N1Cc1cccc(C(=O)NCC2CCN(C)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.44
ROCK2 O75116 12/20 0.42
CDK1 P06493 1/20 0.42
CCNB1 P14635 1/20 0.42
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
ROCK1 Q13464 7/20 0.41
GLS O94925 1/20 0.40
GSK3B P49841 1/20 0.40
DYRK1A Q13627 1/20 0.40
DDR2 Q16832 1/20 0.39
JAK2 O60674 1/20 0.39
MAP4K4 O95819 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25529693 0.90 ROCK2 (0.51) PARP1ROCK2ROCK1
SCHEMBL25528196 0.84 ROCK2 (0.43) PARP1ROCK2ROCK1GLSGSK3B
SCHEMBL25528343 0.84 PARP1 (0.43) PARP1ROCK2CDK1CCNB1CCNA2
SCHEMBL25528200 0.80 ROCK2 (0.40) PARP1ROCK2ROCK1GSK3BMAP4K4
SCHEMBL25531233 0.79 IRAK4 (0.42) PARP1ROCK2ROCK1GSK3B
SCHEMBL25528771 0.79 ROCK2 (0.42) PARP1ROCK2ROCK1
SCHEMBL25528201 0.78 ROCK2 (0.39) PARP1ROCK2ROCK1GSK3BMAP4K4
SCHEMBL25528339 0.78 PARP1 (0.41) PARP1ROCK2ROCK1GLSMAP4K4
SCHEMBL25529692 0.78 ROCK2 (0.52) ROCK2ROCK1
SCHEMBL25528185 0.77 ROCK2 (0.43) ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed