SCHEMBL25528475

SCHEMBL25528475

C[C@@H]1C(=O)N(C)c2cc(-c3ccncc3)ccc2C(=O)N1Cc1cc(F)cc(C(=O)NCC2CC(O)C2)c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 7/20 0.36
AURKA O14965 1/20 0.35
ROCK2 O75116 6/20 0.35
ROCK1 Q13464 3/20 0.35
USP30 Q70CQ3 1/20 0.33
MAP4K4 O95819 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25531283 1.00 CACNA1H (0.36) CACNA1HAURKAROCK2ROCK1USP30
SCHEMBL25528470 0.93 AURKA (0.37) CACNA1HAURKAROCK2ROCK1USP30
SCHEMBL25528185 0.90 ROCK2 (0.43) AURKAROCK2ROCK1
SCHEMBL25529068 0.90 ROCK2 (0.43) AURKAROCK2ROCK1
SCHEMBL25528626 0.90 CCR3 (0.37) AURKAROCK2ROCK1MAP4K4
SCHEMBL25528621 0.89 CACNA1H (0.36) CACNA1HAURKAROCK2ROCK1USP30
SCHEMBL25528945 0.89 CACNA1H (0.36) CACNA1HAURKAROCK2ROCK1USP30
SCHEMBL25528922 0.89 CACNA1H (0.35) CACNA1HAURKAROCK2ROCK1USP30
SCHEMBL25532518 0.89 CACNA1H (0.36) CACNA1HAURKAROCK2ROCK1USP30
SCHEMBL25531296 0.89 ROCK2 (0.33) CACNA1HAURKAROCK2ROCK1USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed