SCHEMBL2552976

SCHEMBL2552976

O=C(CN1C[C@@H]2C[C@H]1CO2)Nc1nc2cc(F)c(Sc3nnc4ccc(C5CC5)nn34)cc2s1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MET P08581 16/20 0.46
CYP3A4 P08684 5/20 0.38
WNT1 P04628 2/20 0.37
GSK3B P49841 2/20 0.37
DYRK1A Q13627 2/20 0.37
WNT3A P56704 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2553465 0.89 MET (0.53) METCYP3A4
SCHEMBL2576776 0.84 MET (0.54) METCYP3A4
SCHEMBL2550322 0.83 MET (0.57) METCYP3A4
SCHEMBL2552274 0.83 MET (0.49) METCYP3A4
SCHEMBL2554270 0.81 MET (0.63) METCYP3A4
SCHEMBL3720726 0.75 MET (0.49) METCYP3A4
SCHEMBL3722617 0.74 MET (0.50) METCYP3A4
SCHEMBL2553888 0.74 MET (0.57) METCYP3A4
SCHEMBL2576078 0.73 MET (0.59) METCYP3A4
SCHEMBL2552619 0.73 MET (0.54) METCYP3A4DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011121223-A1 6-(ALKYL- OR CYCLOALKYL-TRIAZOLOPYRIDAZINE-SULFANYL) BENZOTHIAZOLE DERIVATIVES: PREPARATION, APPLICATION AS MEDICAMENTS AND USE AS MET INHIBITORS SANOFI-AVENTIS (FR) 2011-10-06 WO claimed
WO-2011121223-A1 6-(ALKYL- OR CYCLOALKYL-TRIAZOLOPYRIDAZINE-SULFANYL) BENZOTHIAZOLE DERIVATIVES: PREPARATION, APPLICATION AS MEDICAMENTS AND USE AS MET INHIBITORS SANOFI-AVENTIS (FR) 2011-10-06 WO disclosed