SCHEMBL255440

SCHEMBL255440

COC(=O)[C@H](NC(=O)c1ccc(-c2ccc(N)cc2)cc1)[C@@H](C)O

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 4/20 0.48
TAS1R1 Q7RTX1 4/20 0.48
CA2 P00918 2/20 0.47
CA1 P00915 1/20 0.47
ERAP2 Q6P179 1/20 0.47
LNPEP Q9UIQ6 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
HPGDS O60760 1/20 0.43
SCN1A P35498 1/20 0.42
SCN2A Q99250 1/20 0.42
SCN3A Q9NY46 1/20 0.42
ADRB2 P07550 1/20 0.41
ADRB1 P08588 1/20 0.41
ADRB3 P13945 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
F10 P00742 1/20 0.39
PRSS1 P07477 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL255181 1.00 TAS1R3 (0.48) TAS1R3TAS1R1CA2CA1ERAP2
SCHEMBL1761476 0.90 TAS1R3 (0.59) TAS1R3TAS1R1CA2CA1NPC1
SCHEMBL20299859 0.88 TAS1R3 (0.45) TAS1R3TAS1R1CA2CA1ERAP2
SCHEMBL19262693 0.88 TAS1R3 (0.45) TAS1R3TAS1R1CA2CA1ERAP2
SCHEMBL19262856 0.88 TAS1R3 (0.45) TAS1R3TAS1R1CA2CA1ERAP2
SCHEMBL10272817 0.88 LMNA (0.48) CA2CA1ERAP2NPC1RAB9A
SCHEMBL12055633 0.87 NPC1 (0.54) TAS1R3TAS1R1CA2CA1LNPEP
SCHEMBL1109093 0.87 NPC1 (0.54) TAS1R3TAS1R1CA2CA1LNPEP
SCHEMBL15235727 0.85 TAS1R3 (0.43) TAS1R3TAS1R1CA2CA1ERAP2
SCHEMBL15235725 0.85 TAS1R3 (0.43) TAS1R3TAS1R1CA2CA1ERAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012031298-A2 ETHYNYLBENZENE DERIVATIVES DUKE UNIVERSITY (US) 2012-03-08 WO disclosed