SCHEMBL25547740

SCHEMBL25547740

C1=C(c2cc3ccccc3cn2)CCC2(C1)OCCO2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.52
BTK Q06187 2/20 0.40
NPC1 O15118 3/20 0.37
CYP1A2 P05177 2/20 0.37
KDM4E B2RXH2 2/20 0.37
CASP3 P42574 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
SUV39H2 Q9H5I1 2/20 0.36
RAB9A P51151 2/20 0.35
TBK1 Q9UHD2 2/20 0.35
IKBKE Q14164 1/20 0.35
NPY5R Q15761 1/20 0.34
GRM4 Q14833 1/20 0.34
CYP2A6 P11509 1/20 0.33
PDPK1 O15530 1/20 0.33
MIF P14174 1/20 0.30
HCRTR1 O43613 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL746391 0.77 KDM4E (0.38) TDP1BTKNPC1CYP1A2KDM4E
SCHEMBL25190263 0.77 RAB9A (0.41) TDP1NPC1CYP1A2KDM4ESUV39H2
SCHEMBL20010856 0.76 TBK1 (0.43) TDP1CYP1A2KDM4ESUV39H2TBK1
SCHEMBL20428739 0.75 CCR1 (0.42) BTKKDM4ESUV39H2TBK1IKBKE
SCHEMBL16660952 0.75 IKBKE (0.34) BTKSUV39H2TBK1IKBKE
SCHEMBL25198156 0.75 HDAC4 (0.35) BTKCASP3SENP8SENP7SENP6
SCHEMBL6269678 0.74 P4HTM (0.40) NPC1CYP1A2RAB9AALDH1A1GAA
SCHEMBL629835 0.74 PIK3CD (0.36) BTKSUV39H2TBK1IKBKE
SCHEMBL16680799 0.73 PIK3CA (0.37) BTKSUV39H2TBK1IKBKE
SCHEMBL12208682 0.73 IKBKE (0.41) TDP1NPC1CYP1A2KDM4ESUV39H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023081666-A1 COMPOUNDS AS CCR2 MODULATORS ARIA PHARMACEUTICALS, INC. (US) 2023-05-11 WO disclosed