SCHEMBL2554784

SCHEMBL2554784

O=Cc1cccc(-c2ccc(F)cc2C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRIM24 O15164 1/20 0.51
TRIM33 Q9UPN9 1/20 0.51
BCL2L1 Q07817 1/20 0.48
BAD Q92934 1/20 0.48
UNG P13051 1/20 0.46
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
DHFR P00374 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
LMNA P02545 1/20 0.44
TTR P02766 1/20 0.44
ALB P02768 1/20 0.44
HMGB1 P09429 1/20 0.44
HPGD P15428 1/20 0.44
CXCL12 P48061 1/20 0.44
KMT2A Q03164 1/20 0.44
HIF1A Q16665 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2562602 0.88 TRIM24 (0.51) TRIM24TRIM33BCL2L1BADUNG
SCHEMBL31585756 0.84 DCLRE1B (0.53) KDM4EMEN1USP2ALDH1A1DHFR
SCHEMBL17796982 0.84 DCLRE1B (0.53) KDM4EMEN1USP2ALDH1A1DHFR
SCHEMBL2560064 0.83 HSD17B10 (0.49) KDM4EMEN1USP2ALDH1A1DHFR
SCHEMBL2561114 0.82 TRIM24 (0.51) TRIM24TRIM33UNGKDM4EMEN1
SCHEMBL6715008 0.81 TRIM24 (0.57) TRIM24TRIM33BCL2L1BADUNG
SCHEMBL29952773 0.81 TRIM24 (0.57) TRIM24TRIM33BCL2L1BADUNG
SCHEMBL31585949 0.81 FOLH1 (0.57) KDM4EMEN1USP2ALDH1A1DHFR
SCHEMBL17796951 0.81 FOLH1 (0.57) KDM4EMEN1USP2ALDH1A1DHFR
SCHEMBL2557327 0.79 SMN1; SMN2 (0.62) TRIM24TRIM33UNGKDM4EGPR35

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11225655-B2 Bi-functional complexes and methods for making and using such complexes NUEVOLUTION A/S (DK) 2022-01-18 US disclosed
EP-3540059-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2019-09-18 EP disclosed
EP-2558577-B1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION AS (DK) 2018-12-12 EP disclosed
US-20130281324-A1 BI-FUNCTINAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2013-10-24 US disclosed
EP-2558577-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES Nuevolution A/S (DK) 2013-02-20 EP disclosed
WO-2011127933-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2011-10-20 WO disclosed